PDB Entry - 8J5X

(Status - Released)

Summary information:

Title: The crystal structure of TrkA(G595R) kinase in complex with N-(3-cyclopropyl-5-((4-methylpiperazin-1-yl)methyl)phenyl)-4^6-methyl-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide

PDB DOI: https://doi.org/10.2210/pdb8j5x/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.3c00899

Entry authors: Zhang, Z.M., Wang, Y.J.

Initial deposition on: 24 April 2023

Initial release on: 20 September 2023

Latest revision on: 11 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (mmCIF)

Validation report (PDF)

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