PDB Entry - 8FH4

(Status - Released)

Summary information:

Title: Crystal structure of HPK1 kinase domain T165E,S171E phosphomimetic mutant in complex with 3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undec-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile

PDB DOI: https://doi.org/10.2210/pdb8fh4/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.2c02038

Entry authors: McTigue, M., Johnson, E., Cronin, C.

Initial deposition on: 13 December 2022

Initial release on: 5 April 2023

Latest revision on: 25 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (mmCIF)

Validation report (XML)

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