PDB Entry - 6UF0

(Status - Released)

Summary information:

Title: Crystal structure of N-(4-((4-methoxy-N-(2,2,2-trifluoroethyl)phenyl)sulfonamido)isoquinolin-1-yl)-N-((4-methoxyphenyl)sulfonyl)glycine bound to human Keap1 Kelch domain

PDB DOI: https://doi.org/10.2210/pdb6uf0/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.9b01074

Entry authors: Lazzara, P.R., David, B.P., Ankireddy, A., Richardson, B.G., Dye, K., Ratia, K.M., Reddy, S.P., Moore, T.W.

Initial deposition on: 23 September 2019

Initial release on: 18 December 2019

Latest revision on: 11 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (XML)

Validation report (PDF)

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