PDB Entry - 5VP0
(Status - Released)Summary information:
Title: Discovery of Clinical Candidate N-{(1S)-1-[3-Fluoro-4-(trifluoromethoxy)phenyl]-2-methoxyethyl}-7-methoxy-2-oxo-2,3-dihydropyrido[2,3-b]pyrazine-4(1H)-carboxamide (TAK-915), A Highly Potent, Selective, and Brain-Penetrating Phosphodiesterase 2A Inhibitor for the Treatment of Cognitive Disorders
PDB DOI: https://doi.org/10.2210/pdb5vp0/pdb
Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.7b00807
Entry authors: Hoffman, I.D.
Initial deposition on: 3 May 2017
Initial release on: 23 August 2017
Latest revision on: 13 March 2024
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Structure coordinates (PDB)
X-ray diffraction data (PDBx/mmCIF)
Validation report (mmCIF)
Validation report (XML)
Validation report (PDF)
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