PDB Entry - 5TO8

(Status - Released)

Summary information:

Title: Selectivity switch between FAK and Pyk2: Macrocyclization of FAK inhibitors improves Pyk2 potency

PDB DOI: https://doi.org/10.2210/pdb5to8/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2016.10.092

Entry authors: Newby, Z.E.

Initial deposition on: 17 October 2016

Initial release on: 21 December 2016

Latest revision on: 6 March 2024

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Structure coordinates (PDB)

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