PDB Entry - 5EK9

(Status - Released)

Summary information:

Title: Crystal structure of the second bromodomain of human BRD2 in complex with a tetrahydroquinoline inhibitor

PDB DOI: https://doi.org/10.2210/pdb5ek9/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmc.2017.10.042

Entry authors: Tallant, C., Slavish, P.J., Siejka, P., Bharatham, N., Shadrick, W.R., Chai, S., Young, B.M., Boyd, V.A., Heroven, C., Picaud, S., Fedorov, O., Chen, T., Lee, R.E., Guy, R.K., Shelat, A.A., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Bountra, C., Knapp, S., Structural Genomics Consortium (SGC)

Initial deposition on: 3 November 2015

Initial release on: 16 November 2016

Latest revision on: 8 May 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

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