PDB Entry - 4X7K
(Status - Released)Summary information:
Title: Co-crystal Structure of PERK bound to 4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3H-pyrazol-3-one inhibitor
PDB DOI: https://doi.org/10.2210/pdb4x7k/pdb
Primary publication DOI: https://doi.org/10.1021/jm5017494
Entry authors: Shaffer, P.L., Long, A.M., Chen, H.
Initial deposition on: 9 December 2014
Initial release on: 28 January 2015
Latest revision on: 27 September 2023
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Structure coordinates (PDBML)
Structure coordinates (PDB)
X-ray diffraction data (PDBx/mmCIF)
Validation report (XML)
Validation report (mmCIF)
Validation report (PDF)
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