PDB Entry - 4AJW

(Status - Released)

Summary information:

Title: Discovery and Optimization of New Benzimidazole- and Benzoxazole-Pyrimidone Selective PI3KBeta Inhibitors for the Treatment of Phosphatase and TENsin homologue (PTEN)-Deficient Cancers

PDB DOI: https://doi.org/10.2210/pdb4ajw/pdb

Primary publication DOI: https://doi.org/10.1021/JM300241B

Entry authors: Certal, V., Halley, F., Virone-Oddos, A., Delorme, C., Karlsson, A., Rak, A., Thompson, F., Filoche-Romme, B., El-Ahmad, Y., Carry, J.C., Abecassis, P.Y., Lejeune, P., Bonnevaux, H., Nicolas, J.P., Bertrand, T., Marquette, J.P., Michot, N., Benard, T., Below, P., Vade, I., Chatreaux, F., Lebourg, G., Pilorge, F., Angouillant-Boniface, O., Louboutin, A., Lengauer, C., Schio, L.

Initial deposition on: 20 February 2012

Initial release on: 16 May 2012

Latest revision on: 20 December 2023

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