PDB Entry - 4MR3

(Status - Released)

Summary information:

Title: Crystal Structure of the first bromodomain of human BRD4 in complex with a quinazolinone ligand (RVX-OH)

PDB DOI: https://doi.org/10.2210/pdb4mr3/pdb

Primary publication DOI: https://doi.org/10.1073/pnas.1310658110

Entry authors: Filippakopoulos, P., Picaud, S., Felletar, I., Martin, S., Fedorov, O., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Weigelt, J., Bountra, C., Knapp, S., Structural Genomics Consortium (SGC)

Initial deposition on: 17 September 2013

Initial release on: 27 November 2013

Latest revision on: 12 March 2025

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

Validation report (mmCIF)

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